[H-3] Palbociclib

[H-3] Palbociclib

In stock and ready to ship within 1–2 weeks

Amount

Key Facts

Catalog Number
RCTT2180
CAS Registry Number
571190-30-2
Molecular formula
C24H29N7O2
Molecular weight
447.53 g/mol
Specific Activity Range
50-100 Ci/mmol (1850-3700 GBq/mmol)
Concentration
1.0 mCi/ml (37 MBq/ml) in ethanol.

Description

Orally active and selective CDK4 and CDK6 inhibitor. Has potent antiproliferative activity and induces cell cycle arrest in cancer cells.

Technical Specifications

Product name
[H-3] Palbociclib
Catalog Number
RCTT2180
CAS Registry Number
571190-30-2
Molecular formula
C24H29N7O2
Molecular weight
447.53 g/mol
Concentration
1.0 mCi/ml (37 MBq/ml) in ethanol.
Radiochemical purity
The radiochemical purity after purification was determined to be >97%.
Specific Activity Range
50-100 Ci/mmol (1850-3700 GBq/mmol)
Shipping
Shipped on dry ice.

Storage & Stability

The initial rate of degradation of this compound, stored as received, at temperatures below -60 °C in the dark, is currently under investigation. The decomposition of the compound is not linear or related to isotope half-life. Deviations of different lots may occur.

Safety & Compliance

The compound was isolated from the HPLC eluent under neutral conditions by solid phase extraction. The mass spectrum is consistent with the proposed structure and a non-labeled reference; the HPLC retention time is consistent with a non-labeled reference. Actual position of labels not verified. For research and development use only, not for use in humans.

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